What is the catalog number for TAK-243?

The catalog number for TAK-243 is orb1307707.

What sizes are available for TAK-243?

TAK-243 is available in the following size(s): 1 mg, 2 mg, 5 mg, 1 ml x 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg.

How many pack sizes does TAK-243 come in?

TAK-243 is available in 8 different pack sizes.

TAK-243 is currently made to order / not held in immediate stock. Contact us for lead time.

TAK-243

TAK-243 (MLN7243) is a potent and selective inhibitor of the ubiquitin-activating enzyme (UAE/UBA1) with an IC50 of 1 nM. It effectively blocks global protein ubiquitination, disrupting key cellular signaling pathways. This mechanism underlies its observed pro-apoptotic and antitumor effects in both in vitro and in vivo cancer research models.

Product Specifications

CAS Number

1450833-55-2

Product Name Alternative

Apoptosis, E3Enzyme, E2 conjugating enzyme, E2 Enzyme, E2Enzyme, E3 Enzyme, E3 ligating enzyme, E1 activating enzyme, E1 Enzyme, E1/E2/E3 Enzyme, E1Enzyme, Inhibitor, inhibit, NF-κB, NFκB, NF-kB, NFkB, MLN 7243, MLN7243, MLN-7243, Nuclear factor-kappaB, Nuclear factor-κB, UBA1, Ubiquitin activating enzyme, Ubiquitin conjugating enzyme, Ubiquitin ligase, TAK 243, TAK243, TAK-243