N-desmethyl Enzalutamide
N-desmethyl Enzalutamide is the pharmacologically active primary metabolite of the androgen receptor antagonist Enzalutamide. It exhibits comparable potency and plasma exposure, making it a critical subject for in vitro binding studies and in vivo pharmacological research on prostate cancer models.
Product Specifications
CAS Number
1242137-16-1
Product Name Alternative
AndrogenReceptor, Androgen-receptor, Androgen Receptor, Androgen receptor, Inhibitor, N desmethyl Enzalutamide, inhibit, N-desmethyl MDV3100, N-desmethyl MDV-3100, Ndesmethyl Enzalutamide, N-desmethyl Enzalutamide, N-desmethyl MDV 3100
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Purity
99.62% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.44 mM) ; DMSO:50 mg/mL (111.01 mM)
Smiles
CC1 (C) N (C (=S) N (C1=O) c1ccc (C#N) c (c1) C (F) (F) F) c1ccc (C (N) =O) c (F) c1
Molecular Formula
C20H14F4N4O2S
Molecular Weight
450.41
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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