What is the catalog number for I-BET151?

The catalog number for I-BET151 is orb1306440.

What sizes are available for I-BET151?

I-BET151 is available in the following size(s): 1 mg, 2 mg, 5 mg, 1 ml x 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg, 500 mg.

How many pack sizes does I-BET151 come in?

I-BET151 is available in 9 different pack sizes.

Is I-BET151 in stock?

I-BET151 is currently made to order / not held in immediate stock. Contact us for lead time.

I-BET151

I-BET151 (GSK1210151A) is a potent and selective small-molecule inhibitor of the BET bromodomain proteins BRD2, BRD3, and BRD4, with reported IC50 values of 0.5, 0.25, and 0.79 μM, respectively, in biochemical assays. It is widely used as a chemical probe in cancer, immunology, and inflammation research, demonstrating activity in both cellular studies and in vivo animal models of leukemia and myeloma.

Product Specifications

CAS Number

1300031-49-5

Product Name Alternative

BRD3, BRD2, BRD4, BET, bromodomain, EpigeneticReaderDomain, Epigenetic Reader Domain, I BET151, I-BET 151, IBET151, I-BET151, I-BET-151, GSK1210151A, Inhibitor, inhibit