Cerlapirdine
Cerlapirdine (PF-05212365) is a potent and selective full antagonist of the 5-HT6 receptor. It is utilized in preclinical research for cognitive disorders, with studies investigating its effects in both in vitro binding assays and in vivo models relevant to Alzheimer's disease and schizophrenia.
Product Specifications
CAS Number
925448-93-7
Product Name Alternative
Inhibitor, inhibit, oral, Cerlapirdine, Alzheimer's disease, antagonist, 5HT Receptor, 5-HT Receptor, 5-hydroxytryptamine Receptor, 5HTReceptor, 5-hydroxytryptamine, 5-HT6, SAM 531, SAM531, SAM-531, selective, P -05212365, WAY-262,531, Serotonin Receptor, PF05212365, PF-05212365, PF 05212365
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.60% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.88 mM) ; DMSO:38 mg/mL (92.8 mM)
Smiles
S (=O) (=O) (C=1C=2C (NN1) =CC=C (OCCCN (C) C) C2) C=3C4=C (C=CC3) C=CC=C4
Molecular Formula
C22H23N3O3S
Molecular Weight
409.5
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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