EST73502
EST73502 is a bifunctional small molecule exhibiting μ-opioid receptor agonism (Ki = 64 nM) and σ1 receptor antagonism (Ki = 118 nM) . It demonstrates antinociceptive properties in vivo, making it a useful research tool for investigating pain mechanisms and dual-target analgesic strategies in both cellular and animal models.
Product Specifications
CAS Number
2307458-82-6
Product Name Alternative
2307458-82-6, EST73502, EST-73502, EST73502 HCl, Opioid Receptor, OpioidReceptor, δ-opioid receptor, μ-opioid receptor
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Purity
97.66% (May vary between batches)
Solubility
DMSO:50 mg/mL (128.57 mM)
Smiles
Cl.CCN1CC2 (CCN (CCc3cc (F) ccc3F) CC2) O[C@H] (C) C1=O
Molecular Formula
C19H27ClF2N2O2
Molecular Weight
388.88
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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