PF-CBP1
PF-CBP1 HCl is a potent and selective bromodomain inhibitor targeting CREBBP (IC50 = 125 nM) and its paralog p300 (IC50 = 363 nM) . This small molecule is a valuable chemical probe for epigenetic research, enabling the study of BET-independent transcriptional regulation in both cellular and in vivo models of cancer and other diseases.
Product Specifications
CAS Number
1962928-21-7
Product Name Alternative
Inhibit, Epigenetic Reader Domain, EpigeneticReaderDomain, Inhibitor, CREB, PF-CBP-1, PF-CBP1, PFCBP1, PF CBP1
Field of Research
Cell Biology, Epigenetics & Chromatin
Purity
99.45% (May vary between batches)
Solubility
DMSO:50 mg/mL (102.33 mM)
Smiles
C (CN1CCOCC1) N2C=3C (N=C2CCC4=CC=C (OCCC) C=C4) =CC (=CC3) C=5C (C) =NOC5C
Molecular Formula
C29H36N4O3
Molecular Weight
488.62
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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