Fezolinetant
Fezolinetant (ESN-364) is a selective neurokinin-3 (NK3) receptor antagonist under investigation for the treatment of vasomotor symptoms associated with menopause. Its mechanism of action has been validated in both in vitro binding assays and in vivo preclinical models of thermoregulation.
Product Specifications
CAS Number
1629229-37-3
Product Name Alternative
Neurokinin Receptor, Neurokinin receptor, Neurokininreceptor, NK3, NK receptor, inhibit, Inhibitor, ESN 364, ESN364, ESN-364, Fezolinetant, Tachykinin receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.62% (May vary between batches)
Solubility
DMSO:10 mg/mL (27.9 mM)
Smiles
C[C@H]1N (CCn2c1nnc2-c1nc (C) ns1) C (=O) c1ccc (F) cc1
Molecular Formula
C16H15FN6OS
Molecular Weight
358.39
Storage Conditions
-20°C
Notes
For research use only.
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