BRD4 Inhibitor-10
BRD4 Inhibitor-10 is a potent and selective small molecule targeting the first bromodomain (BD1) of BRD4 with an IC50 of 8 nM. This compound is a valuable chemical probe for epigenetic research, utilized in vitro to study transcriptional regulation in oncology and inflammation, and has been employed in vivo in preclinical cancer models.
Product Specifications
CAS Number
1660117-38-3
Product Name Alternative
BRD4-BD1, BRD4 Inhibitor 10, BRD4 Inhibitor10, BRD-4 Inhibitor-10, BRD4 Inhibitor-10, inhibit, Inhibitor, EpigeneticReaderDomain, Epigenetic Reader Domain
Field of Research
Epigenetics & Chromatin, Epigenetics & Chromatin; Pharmacology & Drug Discovery
Purity
98.98% (May vary between batches)
Solubility
DMSO:125 mg/mL (291.03 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.31 mM)
Smiles
C[C@@H] (c1ccccc1) n1c (nc2cnc (cc12) C1CCOCC1) -c1cc (C) c (=O) n (C) n1
Molecular Formula
C25H27N5O2
Molecular Weight
429.51
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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