TPA 023
TPA 023 is a potent and selective agonist for GABAA receptors containing α2 and/or α3 subunits, exhibiting binding affinities in the sub-nanomolar range (Ki = 0.19 - 0.41 nM) . This compound is a valuable research tool for investigating the roles of specific GABAA receptor subtypes in anxiety, sedation, and cognitive functions in both in vitro and in vivo studies.
Product Specifications
CAS Number
252977-51-8
Product Name Alternative
GABA Receptor, GABAA, GABAReceptor, Gamma-aminobutyric acid Receptor, Inhibitor, inhibit, TPA 023, TPA023, TPA-023, γ-Aminobutyric acid Receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
99.06% (May vary between batches)
Solubility
DMSO:50 mg/mL (126.44 mM)
Smiles
CCn1ncnc1COc1nn2c (nnc2cc1C (C) (C) C) -c1ccccc1F
Molecular Formula
C20H22FN7O
Molecular Weight
395.43
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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