Gαq/11 protein-IN-1
Gαq/11 protein-IN-1 (compound F33) is an inhibitor of Gαq/11 protein with an IC50 value of 9.4 μM. Gαq/11 protein-IN-1 has antitumor activity[1].
Product Specifications
UNSPSC
12352005
Target
Trace Amine-associated Receptor (TAAR)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gαq-11-protein-in-1.html
Solubility
10 mM in DMSO
Smiles
C12=CC=CC=C1C(NC3CCCCC3)=NC(NC4CCNCC4)=N2
Molecular Formula
C19H27N5
Molecular Weight
325.45
References & Citations
[1]Guangjin Fan, et al .Design, synthesis and evaluation of quinazoline derivatives as Gαq/11 proteins inhibitors against uveal melanoma. Bioorg Chem. 2024.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS6407979-01 0.1 mL
AZIN1 (Antizyme Inhibitor 1, Ornithine Decarboxylase Antizyme Inhibitor, OAZI, OAZIN, ODC1L) (MaxLight 550)
Sign In for Pricing
View Details MBS6407979-02 5x 0.1 mL
AZIN1 (Antizyme Inhibitor 1, Ornithine Decarboxylase Antizyme Inhibitor, OAZI, OAZIN, ODC1L) (MaxLight 550)
Sign In for Pricing
View Details