Gαq/11 protein-IN-1
Gαq/11 protein-IN-1 (compound F33) is an inhibitor of Gαq/11 protein with an IC50 value of 9.4 μM. Gαq/11 protein-IN-1 has antitumor activity[1].
Product Specifications
UNSPSC
12352005
Target
Trace Amine-associated Receptor (TAAR)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gαq-11-protein-in-1.html
Solubility
10 mM in DMSO
Smiles
C12=CC=CC=C1C(NC3CCCCC3)=NC(NC4CCNCC4)=N2
Molecular Formula
C19H27N5
Molecular Weight
325.45
References & Citations
[1]Guangjin Fan, et al .Design, synthesis and evaluation of quinazoline derivatives as Gαq/11 proteins inhibitors against uveal melanoma. Bioorg Chem. 2024.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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