I-BET762
Molibresib (GSK525762) is a potent and selective BET bromodomain inhibitor with an IC50 of approximately 35 nM. It is widely used in cancer research, demonstrating activity in both in vitro assays and in vivo models for studying oncology and transcriptional regulation.
Product Specifications
CAS Number
1260907-17-2
Product Name Alternative
GSK525762
Field of Research
Epigenetics & Chromatin, Immunology & Inflammation
Purity
>98%
Bioactivity
BET Bromodomain inhibitor; Suppresses Myc transcription
Form
Powder
Solubility
Soluble in DMSO (up to at least 25 mg/ml) or in Ethanol (up to at least 25 mg/ml)
Smiles
CCNC (=O) C[C@@H]1N=C (c2ccc (Cl) cc2) c2cc (OC) ccc2-n2c (C) nnc12
Molecular Formula
C22H22ClN5O2
Molecular Weight
423.90
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
(4S) - 6- (4-Chlorophenyl) -N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide
Available Sizes
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