Enzastaurin

Enzastaurin (LY317615) is a potent and selective PKCβ inhibitor with an IC50 of 6 nM, exhibiting 6-20 fold selectivity over PKCα, γ, and ε isoforms. It has been widely used in preclinical cancer research, including in vitro cell studies and in vivo tumor models, to investigate angiogenesis and cell signaling pathways.

Product Specifications

CAS Number

170364-57-5

Product Name Alternative

LY-317615

Field of Research

Cell Biology, Neuroscience

Purity

>98%

Bioactivity

PKC inhibitor

Form

Powder

Solubility

Soluble in DMSO (up to 7 mg/ml with warming)

Smiles

O=C1C (C=2C=3C (N (C2) C4CCN (CC5=CC=CC=N5) CC4) =CC=CC3) =C (C (=O) N1) C=6C=7C (N (C) C6) =CC=CC7

Molecular Formula

C32H29N5O2

Molecular Weight

515.61

Storage Conditions

-20°C

Notes

For research use only.

Other Product Names

3- (1-Methyl-1H-indol-3-yl) -4-[1-[1- (2-pyridinylmethyl) -4-piperidinyl]-1H-indol-3-yl]-1H-pyrrole-2,5-dione

Available Sizes

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