ASP-9521
ASP-9521 is a potent, selective, and orally bioavailable indole-based inhibitor targeting AKR1C3, demonstrating an IC50 of 11 nM against the human enzyme. It is a valuable research tool for investigating conditions like castration-resistant prostate cancer and hormone-dependent malignancies in both in vitro and in vivo models.
Product Specifications
CAS Number
1126084-37-4
Product Name Alternative
ASP 9521, ASP9521, ASP-9521, AKR1C3, inhibit, Inhibitor
Field of Research
Metabolism Research
Purity
95.11% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (6.05 mM) ; DMSO:60 mg/mL (181.59 mM)
Smiles
COc1ccc2[nH]c (cc2c1) C (=O) N1CCC (CC (C) (C) O) CC1
Molecular Formula
C19H26N2O3
Molecular Weight
330.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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