Ralinepag
Ralinepag (APD811) is a potent, orally active non-prostanoid IP receptor agonist, exhibiting EC50 values of 8.5 nM (human IP), 530 nM (rat IP), and 850 nM (human DP1) . It is a research tool used in vitro and in vivo to study pulmonary arterial hypertension and other IP receptor-mediated pathways.
Product Specifications
CAS Number
1187856-49-0
Product Name Alternative
APD811, APD-811, APD 811, Inhibitor, inhibit, Prostaglandin Receptor, ProstaglandinReceptor, Prostacyclin receptor, Ralinepag
Field of Research
Immunology & Inflammation, Pharmacology & Drug Discovery
Purity
99.41% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.63 mM) ; DMSO:55 mg/mL (127.34 mM)
Smiles
OC (=O) COC[C@H]1CC[C@H] (COC (=O) N (c2ccccc2) c2ccc (Cl) cc2) CC1
Molecular Formula
C23H26ClNO5
Molecular Weight
431.91
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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