GSK2830371
GSK 2830371 is a potent, cell-permeable allosteric inhibitor of the Wip1 phosphatase, exhibiting an IC50 of 6 nM. It is utilized in cancer research to study p53-dependent pathways and has demonstrated antitumor activity in preclinical in vivo models of various cancers.
Product Specifications
CAS Number
1404456-53-6
Product Name Alternative
GSK2830371, GSK-2830371, GSK 2830371, inhibit, Inhibitor, Wip1 phosphatase, Phosphatase
Field of Research
Metabolism Research
Purity
>97%
Bioactivity
WIP1 phosphatase inhibitor
Form
Powder
Solubility
Soluble in DMSO (up to at least 25 mg/ml)
Smiles
Cc1ncc (Cl) cc1NCc1ccc (s1) C (=O) N[C@@H] (CC1CCCC1) C (=O) NC1CC1
Molecular Formula
C23H29ClN4O2S
Molecular Weight
461.0
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
5-[[ (5-Chloro-2-methylpyridin-3-yl) amino]methyl]-N-[ (2S) -3-cyclopentyl-1- (cyclopropylamino) -1-oxopropan-2-yl]thiophene-2-carboxamide
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