TG 4-155
TG4-155 is a potent and selective brain-penetrant antagonist of the EP2 receptor (KB = 2.4 nM), exhibiting >1000-fold selectivity over EP4 and other off-targets. This profile makes it a valuable research tool for investigating EP2-mediated neuroinflammation, neurodegeneration, and pain in both cellular and animal models.
Product Specifications
CAS Number
1164462-05-8
Product Name Alternative
Inhibitor, EP2, inhibit, TG4 155, TG4155, TG-4-155, TG4-155, Prostaglandin Receptor, ProstaglandinReceptor
Field of Research
Immunology & Inflammation, Pharmacology & Drug Discovery
Purity
>98%
Bioactivity
EP2 receptor antagonist
Form
Powder
Solubility
Soluble in DMSO (up to 35 mg/ml) or in Ethanol (up to 10 mg/ml) .
Smiles
COc1cc (\C=C\C (=O) NCCn2c (C) cc3ccccc23) cc (OC) c1OC
Molecular Formula
C23H26N2O4
Molecular Weight
394.47
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
(2E) -N-[2- (2-Methyl-1H-indol-1-yl) ethyl]-3- (3,4,5-trimethoxyphenyl) -2-propenamide
Available Sizes
Frequently Asked Questions
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