EZM 2302
EZM 2302 (GSK3359088) is a potent and orally bioavailable inhibitor of the arginine methyltransferase CARM1, exhibiting an IC50 of 6 nM. This small molecule is a valuable research tool for investigating CARM1's role in transcriptional regulation, cancer biology, and immune function in both cellular and animal studies.
Product Specifications
CAS Number
1628830-21-6
Product Name Alternative
CARM1, Inhibitor, inhibit, HistoneMethyltransferase, Histone Methyltransferase, EZM 2302, EZM2302, EZM-2302, GSK3359088, GSK-3359088, GSK 3359088
Field of Research
Epigenetics & Chromatin
Purity
97.47% (May vary between batches)
Solubility
DMSO:128.8 mg/mL (220.14 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (6.84 mM)
Smiles
CNC[C@@H] (O) COc1ccc (Cl) c (c1) -c1nc (N2CC3 (C2) CCN (CC3) C (=O) OC) c (C) c (n1) -c1c (C) noc1C
Molecular Formula
C29H37ClN6O5
Molecular Weight
585.09
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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