PROTAC ERRα ligand 2
This compound is a potent PROTAC-based inverse agonist of estrogen-related receptor α (ERRα), exhibiting an IC50 of 5.67 nM. It serves as a valuable chemical tool for studying ERRα function and degradation in cancer metabolism and energy homeostasis research, applicable in both cellular and biochemical assays.
Product Specifications
CAS Number
2306388-57-6
Product Name Alternative
Estrogen Receptor, Estrogen Receptor/ERR, EstrogenReceptor, ERR, ERRα, inhibit, Inhibitor, PROTAC ERRa ligand 2, PROTAC ERRalpha ligand 2, PROTAC ERRα ligand 2, PROTAC ERRα ligand2, PROTAC ERRα ligand-2, progestogenReceptor, progestogen Receptor
Field of Research
Metabolism Research
Purity
≥95% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.49 mM) ; DMSO:10 mM
Smiles
COc1cc (\C=C (/C#N) C (O) =O) ccc1OCc1ccc (cc1C (F) (F) F) C (F) (F) F
Molecular Formula
C20H13F6NO4
Molecular Weight
445.31
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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