Sarpogrelate hydrochloride
Sarpogrelate hydrochloride is a selective 5-HT2A/2B receptor antagonist used as an antiplatelet agent for peripheral arterial disease (PAD) research. It demonstrates high affinity for 5-HT2A receptors (Ki = 8.39 nM) and has been shown in clinical studies to improve vascular function and blood flow in PAD patients following long-term oral administration.
Product Specifications
CAS Number
135159-51-2
Product Name Alternative
Vascular, thrombosis, Serotonin Receptor, Sarpogrelate, Sarpogrelate hydrochloride, Sarpogrelate Hydrochloride, inhibit, Inhibitor, MCI 9042, MCI9042, MCI-9042, 5-HT2R, 5HT Receptor, 5-HT Receptor, 5-HT2, 5-HT2A, 5HTReceptor, 5-hydroxytryptamine Receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
99.42% (May vary between batches)
Solubility
DMSO:245 mg/mL (525.78 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.29 mM)
Smiles
Cl.COc1cccc (CCc2ccccc2OCC (CN (C) C) OC (=O) CCC (O) =O) c1
Molecular Formula
C24H32ClNO6
Molecular Weight
465.97
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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