Thioperamide maleate
Thioperamide maleate (MR-12842 maleate) is a potent and selective histamine H3 receptor antagonist, with a Ki of 4.3 nM for receptor binding and 31 nM for inhibiting [3H]histamine synthesis. This compound is widely used in neuroscience research to study H3 receptor function in both in vitro and in vivo models of sleep, cognition, and energy homeostasis.
Product Specifications
CAS Number
148440-81-7
Product Name Alternative
Histamine Receptor, HistamineReceptor, Inhibitor, H3 receptor, inhibit, MR12842, MR-12842, MR12842 Maleate, MR-12842 maleate, MR-12842 Maleate, MR 12842, MR 12842 Maleate, Thioperamide, Thioperamide maleate, Thioperamide Maleate
Field of Research
Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery
Purity
98.48% (May vary between batches)
Solubility
DMSO:55 mg/mL (134.63 mM)
Smiles
OC (=O) \C=C/C (O) =O.S=C (NC1CCCCC1) N1CCC (CC1) c1cnc[nH]1
Molecular Formula
C19H28N4O4S
Molecular Weight
408.52
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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