S1RA
S1RA hydrochloride (E-52862 hydrochloride) is a potent and selective sigma-1 receptor (σ1R) antagonist with a Ki of 17 nM, demonstrating over 1000-fold selectivity versus the σ2R. This tool compound is widely used in preclinical research to investigate σ1R function in models of neuropathic pain, neurodegenerative diseases, and psychiatric disorders.
Product Specifications
CAS Number
1265917-14-3
Product Name Alternative
E-52862 HCl
Field of Research
Neuroscience
Purity
>98%
Bioactivity
Selective sigma-1 antagonist
Form
Powder
Solubility
Soluble in DMSO (up to at least 25 mg/ml)
Smiles
Cl.Cc1cc (OCCN2CCOCC2) nn1-c1ccc2ccccc2c1
Molecular Formula
C20H23N3O2·HCl
Molecular Weight
373.88
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
4-{2-[5-Methyl-1- (napthalen-2-yl) -1H-pyrazol-3-yloxy]ethyl}morpholine hydrochloride
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