Enzalutamide

Enzalutamide (MDV3100) is a potent androgen receptor antagonist (IC50=36 nM in LNCaP cells) used in research for castration-resistant prostate cancer. It induces autophagy and exhibits antitumor activity, with applications in both in vitro mechanistic studies and in vivo xenograft models.

Product Specifications

CAS Number

915087-33-1

Product Name Alternative

MDV3100; ASP-9785

Field of Research

Cell Biology

Purity

>99%

Bioactivity

Androgen receptor antagonist

Form

Powder

Solubility

Soluble in DMSO (up to 25 mg/ml)

Smiles

S=C1N (C (C) (C) C (=O) N1C2=CC (C (F) (F) F) =C (C#N) C=C2) C3=CC (F) =C (C (NC) =O) C=C3

Molecular Formula

C21H16F4N4O2S

Molecular Weight

464.4

Storage Conditions

-20°C

Notes

For research use only.

Other Product Names

4- (3- (4-Cyano-3- (trifluoromethyl) phenyl) -5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl) -2-fluoro-N-methylbenzamide

Available Sizes

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