Elagolix sodium
Elagolix sodium is a potent and selective GnRH receptor antagonist, with reported IC50 and Ki values of 0.25 nM and 3.7 nM, respectively. It is utilized in research to investigate gonadotropin suppression in preclinical models of endometriosis and uterine fibroids, both in vitro and in vivo.
Product Specifications
CAS Number
832720-36-2
Product Name Alternative
Inhibitor, Elagolix, Elagolix sodium, GnRH Receptor, GNRHR, GNRH Receptor, GnRHR, GNRHReceptor, Gonadotropin releasing hormone receptor, NBI56418, NBI-56418, NBI-56418 sodium, NBI 56418, inhibit
Field of Research
Pharmacology & Drug Discovery
Purity
99.71% (May vary between batches)
Solubility
DMSO:27.78 mg/mL (42.51 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.06 mM) ; H2O:50 mg/mL (76.5 mM)
Smiles
[Na+].COc1cccc (c1F) -c1c (C) n (Cc2c (F) cccc2C (F) (F) F) c (=O) n (C[C@H] (NCCCC ([O-]) =O) c2ccccc2) c1=O
Molecular Formula
C32H29F5N3NaO5
Molecular Weight
653.57
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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