SGC-GAK-1
SGC-GAK-1 is a potent and selective small molecule inhibitor of cyclin G-associated kinase (GAK), exhibiting a Ki of 3.1 nM. This compound is a valuable research tool for investigating GAK's role in cellular processes such as viral entry, autophagy, and Parkinson's disease pathology in both in vitro and in vivo models.
Product Specifications
CAS Number
2226517-76-4
Product Name Alternative
Cyclin G-associated kinase (GAK), Inhibitor, inhibit, SGC GAK 1, SGCGAK1, SGC-GAK-1, Serinekinase, threonin kinase, Serine kinase, threoninkinase
Field of Research
Cell Biology, Metabolism Research
Purity
>99%
Bioactivity
Cyclin G Associated Kinase (GAK) inhibitor
Form
Powder
Solubility
Soluble in DMSO (up to at least 25 mg/ml) or in ethanol (up to 10 mg/ml)
Smiles
COc1cc (Nc2ccnc3ccc (Br) cc23) cc (OC) c1OC
Molecular Formula
C18H17BrN2O3
Molecular Weight
389.25
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
6-Bromo-N- (3,4,5-trimethoxyphenyl) quinoline-4-amine
Available Sizes
Frequently Asked Questions
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