TCS-OX2-29
TCS-OX2-29 is a highly selective orexin receptor 2 (OX2R) antagonist with an IC50 of 40 nM, showing over 250-fold selectivity versus the OX1 receptor. This tool compound is valuable for in vitro and in vivo research exploring the physiological roles of orexin signaling in sleep, arousal, and neuropsychiatric disorders.
Product Specifications
CAS Number
372523-75-6
Product Name Alternative
TCS OX2 29, TCS-OX-2-29, TCS-OX2-29, TCSOX229, inhibit, Orexin Receptor (OX Receptor), OXReceptor, OX2, OX Receptor, Hypocretin Receptor, HCRT Receptor, Inhibitor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
99.08% (May vary between batches)
Solubility
DMSO:9 mg/mL (22.64 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.52 mM)
Smiles
COc1cc2CCN (Cc2cc1OC) C (=O) [C@@H] (NCc1ccncc1) C (C) (C) C
Molecular Formula
C23H31N3O3
Molecular Weight
397.51
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog