GSK-1016790A
GSK1016790A is a potent and selective TRPV4 channel agonist, demonstrating an EC50 of 34 nM in choroid plexus cells. This tool compound is widely used in cardiovascular, pulmonary, and renal research, facilitating the study of TRPV4's role in vitro and in animal models of edema, pain, and mechanosensation.
Product Specifications
CAS Number
942206-85-1
Product Name Alternative
CalciumChannel, Calcium Channel, kidney, mTRPV4, HEK, GSK 101, GSK-101, GSK1016790A, GSK-1016790A, hTRPV4, potential, vanilloid, transient, Transient receptor potential channels, TRPVChannel, TRPChannel, TRPV Channel, TRP Channel
Field of Research
Neuroscience
Purity
>98%
Bioactivity
TRPV4 channel activator
Form
Powder
Solubility
Soluble in DMSO (up to 10 mg/ml) .
Smiles
CC (C) C[C@H] (NC (=O) c1cc2ccccc2s1) C (=O) N1CCN (CC1) C (=O) [C@H] (CO) NS (=O) (=O) c1ccc (Cl) cc1Cl
Molecular Formula
C28H32Cl2N4O6S2
Molecular Weight
655.6
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
(N- ((1S) -1-{[4- ((2S) -2-{[ (2,4-Dichlorophenyl) sulfonyl]amino}-3-hydroxypropanoyl) -1-piperazinyl]carbonyl}-3-methylbutyl) -1-benzothiophene-2-carboxamide
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