Nelotanserin
Nelotanserin (APD125) is a potent and selective inverse agonist of the 5-HT2A receptor (IC50 = 1.7 nM), with moderate activity at 5-HT2C and weak activity at 5-HT2B. It is a valuable research tool for investigating serotonin receptor function in neuropharmacology, sleep disorders, and related in vitro and in vivo studies.
Product Specifications
CAS Number
839713-36-9
Product Name Alternative
5HTReceptor, 5HT Receptor, 5-HT, 5-hydroxytryptamine Receptor, 5-HT Receptor, APD125, APD-125, APD 125, Nelotanserin, inhibit, Inhibitor, Serotonin Receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.01% (May vary between batches)
Solubility
DMSO:250 mg/mL (571.77 mM)
Smiles
COc1ccc (NC (=O) Nc2ccc (F) cc2F) cc1-c1c (Br) cnn1C
Molecular Formula
C18H15BrF2N4O2
Molecular Weight
437.24
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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