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ONO-7300243

ONO-7300243 is a potent and selective LPA1 receptor antagonist with an IC50 of 0.16 μM. This small molecule is a valuable research tool for investigating the role of LPA1 signaling in fibrosis, neuropathic pain, and cancer metastasis in both cellular and animal models.

Product Specifications

CAS Number

638132-34-0

Product Name Alternative

Inhibitor, LPLReceptor, LPL Receptor, LPL, LPAReceptor, LPA Receptor, LPA1, inhibit, Lysophospholipid Receptor, ONO 7300243, ONO7300243, ONO-7300243

Field of Research

Pharmacology & Drug Discovery

Purity

99.66% (May vary between batches)

Solubility

DMSO:100 mg/mL (216.66 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (8.67 mM)

Smiles

COc1cc (cc (OC) c1C) C (=O) N (CCCc1ccccc1) Cc1ccc (CC (O) =O) cc1

Molecular Formula

C28H31NO5

Molecular Weight

461.55

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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