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ERGi-USU

NSC-139021 (ERGi-USU) is a selective small molecule inhibitor targeting Rio2 kinase (RIOK2), leading to the suppression of the oncogenic ERG transcription factor. This compound is utilized in research to investigate ERG-driven cancers, such as prostate leukemia, in both cellular and animal models.

Product Specifications

CAS Number

1147-56-4

Product Name Alternative

NSC139021

Purity

>98%

Bioactivity

Highly selective ERG inhibitor

Form

Powder

Solubility

Soluble in DMSO (up to at least 10 mg/ml)

Smiles

Oc1ccc2ccccc2c1N=Nc1nccs1

Molecular Formula

C13H9N3OS

Molecular Weight

255.30

Storage Conditions

-20°C

Notes

For research use only.

Other Product Names

1- (2-Thiazolylazo) -2-naphthol

Available Sizes

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