A2793
A2793 is a dual TASK-1/TRESK inhibitor exhibiting greater potency and selectivity for TRESK (IC50=6.8 μM for mTRESK) over TREK-1 and TALK-1. This compound serves as a useful pharmacological tool for in vitro electrophysiology studies investigating the roles of these K2P channels in pain sensation and neuronal excitability.
Product Specifications
CAS Number
88349-90-0
Product Name Alternative
A2793, A-2793, A 2793, KcsA, Inhibitor, inhibit, pain, TALK-1, TASK-1, Potassium Channel, PotassiumChannel, TRESK
Field of Research
Pharmacology & Drug Discovery
Purity
97.70% (May vary between batches)
Solubility
DMSO:22.5 mg/mL (84.69 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (7.53 mM)
Smiles
CCOC (=O) COC1=CC=C (Cl) C2=CC=CN=C12
Molecular Formula
C13H12ClNO3
Molecular Weight
265.69
Storage Conditions
-20°C
Notes
For research use only.
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