GSK5182
GSK5182 is a potent and selective inverse agonist of estrogen-related receptor γ (ERRγ), exhibiting an IC50 of 79 nM. This small molecule is a valuable research tool for studying ERRγ's role in metabolic regulation, energy homeostasis, and related diseases in both cellular and animal models.
Product Specifications
CAS Number
877387-37-6
Product Name Alternative
Reactive Oxygen Species, ReactiveOxygenSpecies, progestogen Receptor, progestogenReceptor, inhibit, Inhibitor, ERR, ERRγ, GSK 5182, Estrogen Receptor, Estrogen Receptor/ERR, EstrogenReceptor, GSK5182, GSK-5182
Field of Research
Immunology & Inflammation, Metabolism Research, Signal Transduction
Purity
97.63% (May vary between batches)
Solubility
DMSO:80 mg/mL (191.6 mM)
Smiles
C (=C (/CCCO) \C1=CC=CC=C1) (\C2=CC=C (OCCN (C) C) C=C2) /C3=CC=C (O) C=C3
Molecular Formula
C27H31NO3
Molecular Weight
417.54
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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