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SU4984

SU4984 is a reversible, ATP-competitive, and cell-permeable small molecule inhibitor targeting FGFR1. It is utilized in biochemical and cellular assays to study FGFR1 signaling in cancer research and has been applied in both in vitro and in vivo experimental models.

Product Specifications

CAS Number

186610-89-9

Product Name Alternative

IGF1R, Insulin Receptor, insulin, Inhibitor, factor, fibroblast, Fibroblast growth factor receptor, FGFR1, FGFR, growth, inhibit, kinase, Platelet-derived growth factor receptor, cancer, platelet, SU4984, SU-4984, SU 4984, PDGFR, tyrosine

Field of Research

Cardiovascular Research, Signal Transduction

Purity

97.20% (May vary between batches)

Solubility

DMSO:3.34 mg/mL (10.02 mM)

Smiles

O=CN1CCN (CC1) c1ccc (\C=C2/C (=O) Nc3ccccc23) cc1

Molecular Formula

C20H19N3O2

Molecular Weight

333.38

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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