Paltusotine
Paltusotine is an orally bioavailable, nonpeptide small molecule agonist of the somatostatin type 2 (SST2) receptor. It is used in research to investigate the pharmacological control of growth hormone (GH) and insulin-like growth factor 1 (IGF-1) levels, relevant for acromegaly studies in both in vitro and in vivo models.
Product Specifications
CAS Number
2172870-89-0
Product Name Alternative
CRN 00808, CRN00808, CRN-00808, Inhibitor, IGF-1, inhibit, Paltusotine, orally, SSTRs, SSTR, SST2, Somatostatin Receptor
Field of Research
Pharmacology & Drug Discovery
Purity
99.77% (May vary between batches)
Solubility
DMSO:20 mg/mL (43.81 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.38 mM)
Smiles
NC1CCN (CC1) c1c (cnc2ccc (cc12) -c1cccc (C#N) c1O) -c1cc (F) cc (F) c1
Molecular Formula
C27H22F2N4O
Molecular Weight
456.49
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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