THPP-1
THPP-1 is a highly potent, orally bioavailable PDE10A inhibitor with Ki values of 1 nM (human) and 1.3 nM (rat) . This small molecule is a valuable research tool for investigating PDE10A function in neuropsychiatric disorders, enabling both in vitro biochemical assays and in vivo pharmacological studies.
Product Specifications
CAS Number
1257051-63-0
Product Name Alternative
Novel, inhibit, object, PDE10A, Inhibitor, THPP 1, THPP1, THPP-1, SIMA, recognition, Phosphodiesterase (PDE), phosphodiesterase
Field of Research
Metabolism Research
Purity
99.23% (May vary between batches)
Solubility
DMSO:31 mg/mL (66.68 mM)
Smiles
COCCOc1nc (nc2CCN (Cc12) C (=O) c1ncn2ccccc12) -c1ccc (Cl) nc1
Molecular Formula
C23H21ClN6O3
Molecular Weight
464.9
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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