PW0787
PW0787 is a potent and selective GPR52 agonist with an EC50 of 135 nM. It is orally bioavailable and capable of crossing the blood-brain barrier, making it a valuable research tool for investigating GPR52's role in CNS disorders in both in vitro and in vivo models.
Product Specifications
CAS Number
2624131-45-7
Product Name Alternative
Brain-penetrant, behavior, oral, inhibit, Inhibitor, GPR52, psychostimulant, PW 0787, PW0787, PW-0787, selective
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Purity
98.42% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.34 mM) ; DMSO:65 mg/mL (141.18 mM)
Smiles
OCCNC (=O) c1cccc2N (CCc12) c1cc (Cc2cc (F) cc (c2) C (F) (F) F) ncn1
Molecular Formula
C23H20F4N4O2
Molecular Weight
460.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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