LBP1
LBP1 is an orally active and low brain penetrant CB1 receptor agonist. LBP1 exhibits significant anti-allodynic and anti-hyperalgesic effects in rodent models of neuropathic pain[1].
Product Specifications
CAS Number
1050478-18-6
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/lbp1.html
Smiles
O=C(N)CN1CCN(CC2=NC(C3=CN(CC4CCOCC4)C5=C3C=CC=C5Cl)=NO2)CC1
Molecular Formula
C23H29ClN6O3
Molecular Weight
472.97
References & Citations
[1]Adam J M, et al. Low brain penetrant CB1 receptor agonists for the treatment of neuropathic pain[J]. Bioorganic & medicinal chemistry letters, 2012, 22 (8) : 2932-2937.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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