PLX51107
PLX51107 is a potent, selective BET bromodomain inhibitor with low nanomolar affinity for BRD2, BRD3, BRD4, and BRDT. This small molecule is a valuable research tool for investigating BET protein function in oncology, immunology, and inflammation, supporting both in vitro biochemical assays and in vivo preclinical studies.
Product Specifications
CAS Number
1627929-55-8
Product Name Alternative
BET, inhibit, PLX 51107, PLX51107, PLX-51107, Inhibitor, EpigeneticReaderDomain, Epigenetic Reader Domain
Field of Research
Epigenetics & Chromatin
Purity
99.75% (May vary between batches)
Solubility
DMSO:70 mg/mL (159.64 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.56 mM)
Smiles
C[C@@H] (c1ccccn1) n1cc (-c2ccc (cc2) C (O) =O) c2ncc (cc12) -c1c (C) noc1C
Molecular Formula
C26H22N4O3
Molecular Weight
438.48
Storage Conditions
Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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