RS102895
RS102895 is a selective small molecule antagonist of the CCR2 chemokine receptor with an IC50 of 360 nM, demonstrating no appreciable activity against CCR1. It is a valuable research tool for investigating CCR2-mediated pathways in vitro and has been utilized in studies exploring monocyte migration and inflammatory disease models in vivo.
Product Specifications
CAS Number
300815-41-2
Product Name Alternative
RS 102895, RS102895, RS-102895, inhibit, Inhibitor, CC chemokine receptor, CCR, CCR1
Field of Research
Immunology & Inflammation, Infectious Disease & Virology, Pharmacology & Drug Discovery
Purity
97.64% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.12 mM) ; DMSO:15 mg/mL (38.42 mM)
Smiles
O=C1OC2 (C=3C (N1) =CC=CC3) CCN (CCC4=CC=C (C (F) (F) F) C=C4) CC2
Molecular Formula
C21H21F3N2O2
Molecular Weight
390.4
Storage Conditions
Keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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