SAR-100842
SAR-100842 (SAR100842) is a potent, selective, orally available antagonist of the Lysophosphatidic Acid 1 Receptor (LPA1 receptor) with IC50 of 31 nM in β-arrestin assays; demonstrates potential for the treatment of systemic sclerosis and related fibrotic diseases.Other Indication Phase 2 Discontinued.
Product Specifications
CAS Number
1195941-38-8
Product Name Alternative
SAR100842
Purity
>98% (HPLC)
Solubility
DMSO: Soluble (< 1 mg/ml refers to the product slightly soluble or insoluble)
Smiles
O=C (C1 (NC (C2=CC=C (OC) C (OCCC3=CC=CC (C) =C3) =C2) =O) CC4=C (C=CC=C4) C1) O
Molecular Formula
C27H27NO5
Molecular Weight
445.515
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
2-{4-methoxy-3-[2- (3-methylphenyl) ethoxy]benzamido}-2,3-dihydro-1H-indene-2-carboxylic acid
Available Sizes
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