RQ00203078
RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively), exhibits >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1.
Product Specifications
CAS Number
1254205-52-1
Product Name Alternative
RQ-00203078 | RQ 00203078 | RQ00203078
Purity
>98% (HPLC)
Solubility
DMSO: 100 mM
Smiles
O=C (O) C1=CC=C (S (=O) (N (C2=NC=C (C (F) (F) F) C=C2Cl) CC3=CC=C (OC (F) (F) F) C=C3) =O) C=C1
Molecular Formula
C21H13ClF6N2O5S
Molecular Weight
554.85
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
4- (N- (3-chloro-5- (trifluoromethyl) pyridin-2-yl) -N- (4- (trifluoromethoxy) benzyl) sulfamoyl) benzoic acid
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
