GSK1904529A
GSK1904529A is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM, >100-fold more selective for IGF-1R/InsR than Akt1/2, Aurora A/B, B-Raf, CDK2, EGFR etc.
Product Specifications
CAS Number
1089283-49-7
Product Name Alternative
GSK-4529 | GSK1904529a | GSK 1904529 | GSK-1904529a
Purity
>98% (HPLC)
Solubility
DMSO:124 mg/mL (145.54 mM) ; Ethanol:<1 mg/mL (<1 mM) ; Water:<1 mg/mL (<1 mM)
Smiles
O=C (NC1=C (F) C=CC=C1F) C2=CC (C3=C (C4=NC (NC5=CC (CC) =C (N6CCC (N7CCN (S (=O) (C) =O) CC7) CC6) C=C5OC) =NC=C4) N8C=CC=CC8=N3) =CC=C2OC
Molecular Formula
C44H47F2N9O5S
Molecular Weight
851.96
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
N- (2,6-Difluorophenyl) -5-[3-[2-[[5-ethyl-2- (methyloxy) -4-[4-[4- (methylsulfonyl) -1-piperazinyl]-1-piperidinyl]phenyl]amino]-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl]-2- (methyloxy) benzamide
Available Sizes
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