CCG-215022
CCG-215022 (CCG215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively; displays 300-800 fold selectivity against PKA; exhibits improved potency compared with GSK180736A.
Product Specifications
CAS Number
1813527-81-9
Product Name Alternative
CCG215022 | CCG 215022
Purity
>98% (HPLC)
Solubility
DMSO: ≥ 28 mg/mL
Smiles
O=C (C1=C (F) C=CC (C2C (C (NC3=CC=C (NN=C4) C4=C3) =O) =C (C) NC (N2) =O) =C1) NCC5=NC=CC=C5
Molecular Formula
C26H22FN7O3
Molecular Weight
499.4964
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
4- (4-fluoro-3- ((pyridin-2-ylmethyl) carbamoyl) phenyl) -N- (1H-indazol-5-yl) -6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
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