AM251
AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also potent GPR55 agonist (EC50 = 39 nM) .
Product Specifications
CAS Number
183232-66-8
Product Name Alternative
AM251 | AM 251 | AM-251
Purity
>98% (HPLC)
Solubility
DMSO: 40 mg/mL (72.04 mM)
Smiles
O=C (C1=NN (C2=CC=C (Cl) C=C2Cl) C (C3=CC=C (I) C=C3) =C1C) NN4CCCCC4
Molecular Formula
C22H21Cl2IN4O
Molecular Weight
555.24
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
1- (2,4-dichlorophenyl) -5- (4-iodophenyl) -4-methyl-N- (piperidin-1-yl) -1H-pyrazole-3-carboxamide
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