DBET57
DBET57 is a novel BRD4 heterobifunctional small-molecule ligand (PROTAC), exhibits significant and selective degradation of BRD4 BD1 (DC50/5h=500 nM), but is inactive on BRD4 BD2.
Product Specifications
CAS Number
1883863-52-2
Product Name Alternative
DBET57
Purity
>98% (HPLC)
Solubility
DMSO : 250 mg/mL 357.56 mM
Smiles
O=C (NCCNC1=CC=CC (C (N2C (CC3) C (NC3=O) =O) =O) =C1C2=O) C[C@H]4C5=NN=C (C) N5C6=C (C (C) =C (C) S6) C (C7=CC=C (Cl) C=C7) =N4
Molecular Formula
C34H31ClN8O5S
Molecular Weight
699.183
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
2- ((S) -4- (4-chlorophenyl) -2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl) -N- (2- ((2- (2,6-dioxopiperidin-3-yl) -1,3-dioxoisoindolin-4-yl) amino) ethyl) acetamide
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