EPZ005687
EPZ005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM in a cell-free assay, 50-fold selectivity against EZH1 and 500-fold selectivity against 15 other protein methyltransferases.
Product Specifications
CAS Number
1396772-26-1
Purity
>98% (HPLC)
Solubility
DMSO: 2 mg/mL (3.7 mM)
Smiles
CC1=CC (C) =C (CNC (=O) C2=C3C=NN (C4CCCC4) C3=CC (=C2) C2=CC=C (CN3CCOCC3) C=C2) C (=O) N1
Molecular Formula
C32H37N5O3
Molecular Weight
539.67
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Available Sizes
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