GSK-2879552
A potent, selective irreversible inhibitor of LSD1 with Ki app of 1.7 uM; shows good selectivity against LSD2, MAO-A, MAO-B, D-amino acid oxidase and LoxL2; exhibits growth inhibition (EC50=2-240 nM) in sensitive cell lines; orally bioavailable.Lung Cancer Phase 1 Clinical.
Product Specifications
CAS Number
1401966-69-5
Product Name Alternative
GSK2879552
Purity
>98% (HPLC)
Solubility
10 mM in DMSO
Smiles
O=C (O) C1=CC=C (CN2CCC (CN[C@H]3[C@H] (C4=CC=CC=C4) C3) CC2) C=C1
Molecular Formula
C23H28N2O2
Molecular Weight
364.4806
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
Benzoic acid, 4-[[4-[[[ (1R,2S) -2-phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]-
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