CB1-IN-4
CB1-IN-4 is a potent, selective, peripherally restricted cannabinoid-1 (CB1) receptor antagonist with Ki of 0.3 nM, EC50 of 3.0 nM; possess a low probability to cross BBB as a peripherally restricted CB1R antagonist, exhibits significant weight-loss efficacy in DIO mice, also displays 163 clean off-target profiles and potential for treating obesity and the related metabolic syndrome.
Product Specifications
CAS Number
1429239-98-4
Product Name Alternative
DBPR211 | DBPR 211 | DBPR-211 | CB1-IN-1
Field of Research
Neuroscience
Purity
>98% (HPLC)
Solubility
10 mM in DMSO
Smiles
O=C (C1=NN (C2=CC=C (Cl) C=C2Cl) C (C3=CC=C (C#CC4=CC=C (C (F) (F) F) C=C4) S3) =C1CNS (=O) (N5CCCC5) =O) NN6CCCCC6
Molecular Formula
C33H31Cl2F3N6O3S2
Molecular Weight
751.6688
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
1H-Pyrazole-3-carboxamide, 1- (2,4-dichlorophenyl) -N-1-piperidinyl-4-[[ (1-pyrrolidinylsulfonyl) amino]methyl]-5-[5-[2-[4- (trifluoromethyl) phenyl]ethynyl]-2-thienyl]-
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