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ARV-771

ARV-771 is a potent BET degrader (PROTAC) in cellular models of CRPC; potently degrades BRD2/3/4 in 22Rv1 cells with DC50< 5 nM.

Product Specifications

CAS Number

1949837-12-0

Purity

>98% (HPLC)

Molecular Formula

C49H60ClN9O7S2

Molecular Weight

986.6

Storage Conditions

Storage temperature: -20°C. Stability: ≥ 2 years

Notes

For research use only.

Available Sizes

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