BCTC
A highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively; shows selectivity against 63 other receptor, enzyme, transporter, and ion channel targets; orally bioavailable.Pain Preclinical.
Product Specifications
CAS Number
393514-24-4
Product Name Alternative
BCTC
Purity
>98% (HPLC)
Solubility
10 mM in DMSO
Smiles
O=C (N1CCN (C2=NC=CC=C2Cl) CC1) NC3=CC=C (C (C) (C) C) C=C3
Molecular Formula
C20H25ClN4O
Molecular Weight
372.8917
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
1-Piperazinecarboxamide, 4- (3-chloro-2-pyridinyl) -N-[4- (1,1-dimethylethyl) phenyl]-
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