GSK-180736A
A highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM; displays >400-fold selective for GRK2 over both GRK1 and GRK5, with no inhibition on PKA; also inhibits ROCK with IC50 of 0.1 uM.
Product Specifications
CAS Number
817194-38-0
Product Name Alternative
GSK 180736A | GSK180736A
Purity
>98% (HPLC)
Solubility
DMSO: ≥ 30 mg/mL
Smiles
CC1=C (C (NC (=O) N1) C2=CC=C (C=C2) F) C (=O) NC3=CC4=C (C=C3) NN=C4
Molecular Formula
C19H16FN5O2
Molecular Weight
365.3611
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
5-Pyrimidinecarboxamide, 4- (4-fluorophenyl) -1,2,3,4-tetrahydro-N-1H-indazol-5-yl-6-methyl-2-oxo-
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